产品编号 | CFN60026 | |
CAS编号 | 252917-06-9 | |
分子式 = 分子量 | C22H18Cl2N8 = 465.34 | |
产品纯度 | >=98% | |
物理属性 | Powder | |
化合物类型 | Alkaloids | |
植物来源 | ||
ChemFaces的产品在影响因子大于5的优秀和顶级科学期刊中被引用 |
产品名称 | 产品编号 | CAS编号 | 包装 | QQ客服 |
CHIR-99021 (CT99021) | CFN60026 | 252917-06-9 | 1mg | QQ客服:215959384 |
CHIR-99021 (CT99021) | CFN60026 | 252917-06-9 | 5mg | QQ客服:215959384 |
CHIR-99021 (CT99021) | CFN60026 | 252917-06-9 | 10mg | QQ客服:215959384 |
CHIR-99021 (CT99021) | CFN60026 | 252917-06-9 | 20mg | QQ客服:215959384 |
Description: | CHIR-99021 (CT99021) is a GSK-3α and GSK-3β inhibitor with IC50 of 10 nM and 6.7 nM, respectively. CHIR99201 does not exhibit cross-reactivity against cyclin-dependent kinases (CDKs) and shows a 350-fold selectivity toward GSK-3β compared to CDKs. CHIR99021 functions as a Wnt/β-catenin activator and induces autophagy. |
Targets: | GSK-3α/GSK-3β | CDK | Autophagy |
1 mg | 5 mg | 10 mg | 20 mg | 25 mg | |
1 mM | 2.149 mL | 10.7448 mL | 21.4897 mL | 42.9793 mL | 53.7242 mL |
5 mM | 0.4298 mL | 2.149 mL | 4.2979 mL | 8.5959 mL | 10.7448 mL |
10 mM | 0.2149 mL | 1.0745 mL | 2.149 mL | 4.2979 mL | 5.3724 mL |
50 mM | 0.043 mL | 0.2149 mL | 0.4298 mL | 0.8596 mL | 1.0745 mL |
100 mM | 0.0215 mL | 0.1074 mL | 0.2149 mL | 0.4298 mL | 0.5372 mL |
产品名称 | 产品编号 | CAS编号 | 分子式 = 分子量 | 位单 | 联系QQ |
2-O-甲基马兜铃,胡椒内酰胺C; Piperolactam C | CFN97948 | 116064-76-7 | C18H15NO4 = 309.3 | 5mg | QQ客服:2159513211 |
(-)-飞龙掌血烯醇内酯; (-)-Toddanol | CFN92513 | 77715-99-2 | C16H18O5 = 290.3 | 5mg | QQ客服:1413575084 |
25-O-乙基升麻醇-3-O-β-D-吡喃木糖苷; 25-O-ethylcimigenol-3-O-beta-D-xylopyranoside | CFN92379 | 914086-57-0 | C37H60O9 = 648.9 | 5mg | QQ客服:3257982914 |
光甘草醇; Glabrol | CFN93042 | 59870-65-4 | C25H28O4 = 392.49 | 5mg | QQ客服:215959384 |