产品编号 | CFN60026 | |
CAS编号 | 252917-06-9 | |
分子式 = 分子量 | C22H18Cl2N8 = 465.34 | |
产品纯度 | >=98% | |
物理属性 | Powder | |
化合物类型 | Alkaloids | |
植物来源 | ||
ChemFaces的产品在影响因子大于5的优秀和顶级科学期刊中被引用 |
产品名称 | 产品编号 | CAS编号 | 包装 | QQ客服 |
CHIR-99021 (CT99021) | CFN60026 | 252917-06-9 | 1mg | QQ客服:2159513211 |
CHIR-99021 (CT99021) | CFN60026 | 252917-06-9 | 5mg | QQ客服:2159513211 |
CHIR-99021 (CT99021) | CFN60026 | 252917-06-9 | 10mg | QQ客服:2159513211 |
CHIR-99021 (CT99021) | CFN60026 | 252917-06-9 | 20mg | QQ客服:2159513211 |
Description: | CHIR-99021 (CT99021) is a GSK-3α and GSK-3β inhibitor with IC50 of 10 nM and 6.7 nM, respectively. CHIR99201 does not exhibit cross-reactivity against cyclin-dependent kinases (CDKs) and shows a 350-fold selectivity toward GSK-3β compared to CDKs. CHIR99021 functions as a Wnt/β-catenin activator and induces autophagy. |
Targets: | GSK-3α/GSK-3β | CDK | Autophagy |
1 mg | 5 mg | 10 mg | 20 mg | 25 mg | |
1 mM | 2.149 mL | 10.7448 mL | 21.4897 mL | 42.9793 mL | 53.7242 mL |
5 mM | 0.4298 mL | 2.149 mL | 4.2979 mL | 8.5959 mL | 10.7448 mL |
10 mM | 0.2149 mL | 1.0745 mL | 2.149 mL | 4.2979 mL | 5.3724 mL |
50 mM | 0.043 mL | 0.2149 mL | 0.4298 mL | 0.8596 mL | 1.0745 mL |
100 mM | 0.0215 mL | 0.1074 mL | 0.2149 mL | 0.4298 mL | 0.5372 mL |
产品名称 | 产品编号 | CAS编号 | 分子式 = 分子量 | 位单 | 联系QQ |
Daturataturin A; Daturataturin A | CFN99414 | 133360-51-7 | C34H48O10 = 616.8 | 5mg | QQ客服:3257982914 |
QNZ (EVP4593); QNZ (EVP4593) | CFN60177 | 545380-34-5 | C22H20N4O = 356.42 | 5mg | QQ客服:2056216494 |
人参皂苷Rg6; Ginsenoside Rg6 | CFN90565 | 147419-93-0 | C42H70O12 = 766.5 | 5mg | QQ客服:2159513211 |
异鼠李素-3-O-葡萄糖苷; Isorhamnetin-3-O-beta-D-Glucoside | CFN99757 | 5041-82-7 | C22H22O12 = 478.40 | 10mg | QQ客服:3257982914 |