产品编号 | CFN60026 | |
CAS编号 | 252917-06-9 | |
分子式 = 分子量 | C22H18Cl2N8 = 465.34 | |
产品纯度 | >=98% | |
物理属性 | Powder | |
化合物类型 | Alkaloids | |
植物来源 | ||
ChemFaces的产品在影响因子大于5的优秀和顶级科学期刊中被引用 |
产品名称 | 产品编号 | CAS编号 | 包装 | QQ客服 |
CHIR-99021 (CT99021) | CFN60026 | 252917-06-9 | 1mg | QQ客服:2056216494 |
CHIR-99021 (CT99021) | CFN60026 | 252917-06-9 | 5mg | QQ客服:2056216494 |
CHIR-99021 (CT99021) | CFN60026 | 252917-06-9 | 10mg | QQ客服:2056216494 |
CHIR-99021 (CT99021) | CFN60026 | 252917-06-9 | 20mg | QQ客服:2056216494 |
Description: | CHIR-99021 (CT99021) is a GSK-3α and GSK-3β inhibitor with IC50 of 10 nM and 6.7 nM, respectively. CHIR99201 does not exhibit cross-reactivity against cyclin-dependent kinases (CDKs) and shows a 350-fold selectivity toward GSK-3β compared to CDKs. CHIR99021 functions as a Wnt/β-catenin activator and induces autophagy. |
Targets: | GSK-3α/GSK-3β | CDK | Autophagy |
1 mg | 5 mg | 10 mg | 20 mg | 25 mg | |
1 mM | 2.149 mL | 10.7448 mL | 21.4897 mL | 42.9793 mL | 53.7242 mL |
5 mM | 0.4298 mL | 2.149 mL | 4.2979 mL | 8.5959 mL | 10.7448 mL |
10 mM | 0.2149 mL | 1.0745 mL | 2.149 mL | 4.2979 mL | 5.3724 mL |
50 mM | 0.043 mL | 0.2149 mL | 0.4298 mL | 0.8596 mL | 1.0745 mL |
100 mM | 0.0215 mL | 0.1074 mL | 0.2149 mL | 0.4298 mL | 0.5372 mL |
产品名称 | 产品编号 | CAS编号 | 分子式 = 分子量 | 位单 | 联系QQ |
柘树咕吨酮D; Cudraxanthone D | CFN97543 | 96552-41-9 | C24H26O6 = 410.5 | 5mg | QQ客服:1457312923 |
岩茨烯A; Rehmannic acid | CFN97738 | 467-81-2 | C35H52O5 = 552.80 | 5mg | QQ客服:2056216494 |
盐酸槟榔次碱; Arecaidine hydrochloride | CFN93357 | 6018-28-6 | C7H12ClNO2 = 177.6 | 5mg | QQ客服:3257982914 |
刺甘草查尔酮; Echinatin | CFN99520 | 34221-41-5 | C16H14O4 = 270.28 | 20mg | QQ客服:215959384 |