产品编号 | CFN60056 | |
CAS编号 | 915019-65-7 | |
分子式 = 分子量 | C30H23N5O = 469.55 | |
产品纯度 | >=98% | |
物理属性 | Powder | |
化合物类型 | Alkaloids | |
植物来源 | ||
ChemFaces的产品在影响因子大于5的优秀和顶级科学期刊中被引用 |
产品名称 | 产品编号 | CAS编号 | 包装 | QQ客服 |
Dactolisib (BEZ235) | CFN60056 | 915019-65-7 | 1mg | QQ客服:2159513211 |
Dactolisib (BEZ235) | CFN60056 | 915019-65-7 | 5mg | QQ客服:2159513211 |
Dactolisib (BEZ235) | CFN60056 | 915019-65-7 | 10mg | QQ客服:2159513211 |
Dactolisib (BEZ235) | CFN60056 | 915019-65-7 | 20mg | QQ客服:2159513211 |
Description: | Dactolisib (BEZ235, NVP-BEZ235) is a dual ATP-competitive PI3K and mTOR inhibitor for p110α/γ/δ/β and mTOR(p70S6K) with IC50 of 4 nM /5 nM /7 nM /75 nM /6 nM in cell-free assays, respectively. Inhibits ATR with IC50 of 21 nM in 3T3TopBP1-ER cell. Dactolisib induces autophagy and suppresses HIV-1 replication. |
Targets: | PI3K | mTOR | ATR | Autophagy | HIV |
1 mg | 5 mg | 10 mg | 20 mg | 25 mg | |
1 mM | 2.1297 mL | 10.6485 mL | 21.297 mL | 42.594 mL | 53.2425 mL |
5 mM | 0.4259 mL | 2.1297 mL | 4.2594 mL | 8.5188 mL | 10.6485 mL |
10 mM | 0.213 mL | 1.0648 mL | 2.1297 mL | 4.2594 mL | 5.3242 mL |
50 mM | 0.0426 mL | 0.213 mL | 0.4259 mL | 0.8519 mL | 1.0648 mL |
100 mM | 0.0213 mL | 0.1065 mL | 0.213 mL | 0.4259 mL | 0.5324 mL |
产品名称 | 产品编号 | CAS编号 | 分子式 = 分子量 | 位单 | 联系QQ |
黄柏呈; Phellochin | CFN99252 | 115334-04-8 | C31H52O4 = 488.8 | 5mg | QQ客服:1457312923 |
瑞香素; 瑞香内酯; Daphnetin | CFN99952 | 486-35-1 | C9H6O4 = 178.14 | 20mg | QQ客服:215959384 |
Pepluanin A; Pepluanin A | CFN97144 | 670257-89-3 | C43H51NO15 = 821.9 | 5mg | QQ客服:215959384 |
诃子林鞣酸; Chebulinic acid | CFN92296 | 18942-26-2 | C41H32O27 = 956.7 | 20mg | QQ客服:3257982914 |