产品编号 | CFN60010 | |
CAS编号 | 129-56-6 | |
分子式 = 分子量 | C14H8N2O = 220.23 | |
产品纯度 | >=98% | |
物理属性 | Powder | |
化合物类型 | Alkaloids | |
植物来源 | ||
ChemFaces的产品在影响因子大于5的优秀和顶级科学期刊中被引用 |
产品名称 | 产品编号 | CAS编号 | 包装 | QQ客服 |
吡唑蒽酮(SP600125) | CFN60010 | 129-56-6 | 1mg | QQ客服:2159513211 |
吡唑蒽酮(SP600125) | CFN60010 | 129-56-6 | 5mg | QQ客服:2159513211 |
吡唑蒽酮(SP600125) | CFN60010 | 129-56-6 | 10mg | QQ客服:2159513211 |
吡唑蒽酮(SP600125) | CFN60010 | 129-56-6 | 20mg | QQ客服:2159513211 |
Description: | SP600125 is a broad-spectrum JNK inhibitor for JNK1, JNK2 and JNK3 with IC50 of 40 nM, 40 nM and 90 nM in cell-free assays, respectively; 10-fold greater selectivity against MKK4, 25-fold greater selectivity against MKK3, MKK6, PKB, and PKCα, and 100-fold selectivity against ERK2, p38, Chk1, EGFR etc. SP600125 is also a broad‐spectrum inhibitor of serine/threonine kinases including Aurora kinase A,FLT3 and TRKA with of IC50 of 60 nM, 90 nM and 70 nM. SP600125 inhibits autophagy and activates apoptosis. |
Targets: | JNK | JNK1/JNK2/JNK3 | MKK | PKB | PKCα | ERK | EGFR | p38 | TRKA | Autophagy |
1 mg | 5 mg | 10 mg | 20 mg | 25 mg | |
1 mM | 4.5407 mL | 22.7035 mL | 45.4071 mL | 90.8141 mL | 113.5177 mL |
5 mM | 0.9081 mL | 4.5407 mL | 9.0814 mL | 18.1628 mL | 22.7035 mL |
10 mM | 0.4541 mL | 2.2704 mL | 4.5407 mL | 9.0814 mL | 11.3518 mL |
50 mM | 0.0908 mL | 0.4541 mL | 0.9081 mL | 1.8163 mL | 2.2704 mL |
100 mM | 0.0454 mL | 0.227 mL | 0.4541 mL | 0.9081 mL | 1.1352 mL |
产品名称 | 产品编号 | CAS编号 | 分子式 = 分子量 | 位单 | 联系QQ |
报春黄苷; Sinensin | CFN97925 | 28189-90-4 | C21H22O11 = 450.4 | 5mg | QQ客服:1457312923 |
番茄碱; Tomatidine | CFN90632 | 77-59-8 | C27H45NO2 = 415.65 | 20mg | QQ客服:2056216494 |
Leonloside D; Leonloside D | CFN91043 | 20830-84-6 | C59H96O27 = 1237.39 | 5mg | QQ客服:2056216494 |
14,15-二脱氢异埃那胺; 14,15-Didehydroisoeburnamine | CFN98803 | 50838-11-4 | C19H22N2O = 294.4 | 5mg | QQ客服:3257982914 |